AUDINOT, Valérie: search on Z-Library

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1

4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part. II: Synthesis and pharmacological evaluation of oxime and acidic head group structural variations

Cécile Parmenon, Jérôme Guillard, Daniel-Henri Caignard, Nathalie Hennuyer, Bart Staels, Valérie Audinot-Bouchez, Jean-Albert Boutin, Catherine Dacquet, Alain Ktorza, Marie-Claude Viaud-Massuard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 477 KB

english, 2009

2

ChemInform Abstract: Novel Benzopyrano[3,4-c]pyrrole Derivatives as Potent and Selective Dopamine D3 Receptor Antagonists.

Thierry Dubuffet, Adrian Newman-Tancredi, Didier Cussac, Valerie Audinot, Annie Loutz, Mark J. Millan, Gilbert Lavielle

Journal:

Year:

1999

File:

PDF, 32 KB

1999

3

Synthesis of new 8( S )-HETE analogs and their biological evaluation as activators of the PPAR nuclear receptors

Liutkus, Mélanie, Caijo, Frédéric, Girard, Anne-Lise, Ayral, Erwan, Audinot, Valérie, Boutin, Jean A., Renard, Pierre, Caignard, Daniel Henri, Dacquet, Catherine, Ktorza, Alain, Mosset, Paul, Grée, Re

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.14 MB

english, 2010

4

[125I]-S36057: a new and highly potent radioligand for the melanin-concentrating hormone receptor

Valérie Audinot, Chantal Lahaye, Thomas Suply, Philippe Beauverger, Marianne Rodriguez, Jean-Pierre Galizzi, Jean-Luc Fauchère, Jean A Boutin

Journal:

British Journal of Pharmacology

Year:

2001

Language:

english

File:

PDF, 194 KB

english, 2001

5

Molecular pharmacology of the ovine melatonin receptor: comparison with recombinant human MT1 and MT2 receptors

François Mailliet, Valérie Audinot, Benoit Malpaux, Anne Bonnaud, Philippe Delagrange, Martine Migaud, Perry Barrett, Marie-Claude Viaud-Massuard, Daniel Lesieur, François Lefoulon, Pierre Renard, Jea

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 273 KB

english, 2004

6

Inverse Agonist Properties of Antipsychotic Agents at Cloned, Human (h) Serotonin (5-HT)1B and h5-HT1D Receptors

Valérie Audinot, Adrian Newman-Tancredi, Didier Cussac, Mark J Millan

Journal:

Neuropsychopharmacology

Year:

2001

Language:

english

File:

PDF, 190 KB

english, 2001

7

Synthesis and Structure−Affinity−Activity Relationships of Novel Benzofuran Derivatives as MT 2 Melatonin Receptor Selective Ligands

Wallez, Valérie, Durieux-Poissonnier, Sophie, Chavatte, Philippe, Boutin, Jean A., Audinot, Valérie, Nicolas, Jean-Paul, Bennejean, Caroline, Delagrange, Philippe, Renard, Pierre, Lesieur, Daniel

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 139 KB

english, 2002

8

Blockade of NMDA receptors in the nucleus accumbens elicits spontaneous tail-flicks in rats

Mark J. Millan, Valérie Audinot, Prisca Honoré, Karin Bervoets, Sylvie Veiga, Mauricette Brocco

Journal:

European Journal of Pharmacology

Year:

2000

Language:

english

File:

PDF, 204 KB

english, 2000

9

Evidence that dopamine D3 receptors participate in clozapine-induced hypothermia

Mark J. Millan, Valérie Audinot, Christophe Melon, Adrian Newman-Tancredi

Journal:

European Journal of Pharmacology

Year:

1995

Language:

english

File:

PDF, 451 KB

english, 1995

10

Binding profile of the novel 5-HT1B/1D receptor antagonist, [3H]GR 125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

Valérie Audinot, Sonia Lochon, Adrian Newman-Tancredi, Gilbert Lavielle, Mark J Millan

Journal:

European Journal of Pharmacology

Year:

1997

Language:

english

File:

PDF, 282 KB

english, 1997

11

Synthesis of 3-phenylnaphthalenic derivatives as new selective MT2 melatoninergic ligands

Sophie Poissonnier-Durieux, Mohamed Ettaoussi, Basile Pérès, Jean A. Boutin, Valérie Audinot, Caroline Bennejean, Philippe Delagrange, Daniel Henri Caignard, Pierre Renard, Pascal Berthelot, Daniel Le

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 253 KB

english, 2008

12

Ligand modulation of [35S]GTPγS binding at human α2A, α2B and α2C adrenoceptors

Valérie Audinot, Nelly Fabry, Jean-Paul Nicolas, Philippe Beauverger, Adrian Newman-Tancredi, Mark J Millan, Anne Try, Frédéric Bornancin, Emmanuel Canet, Jean A Boutin

Journal:

Cellular Signalling

Year:

2002

Language:

english

File:

PDF, 207 KB

english, 2002

13

S 14297, a novel selective ligand at cloned human dopamine D3 receptors, blocks 7-OH-DPAT-induced hypothermia in rats

Mark J. Millan, Valérie Audinot, Jean-Michel Rivet, Alain Gobert, Joël Vian, Jean-François Prost, Michael Spedding, Jean-Louis Peglion

Journal:

European Journal of Pharmacology

Year:

1994

Language:

english

File:

PDF, 272 KB

english, 1994

14

Effect of Oxime Ether Incorporation in Acyl Indole Derivatives on PPAR Subtype Selectivity

Le Naour, Morgan, Leclerc, Veronique, Farce, Amaury, Caignard, Daniel-Henri, Hennuyer, Nathalie, Staels, Bart, Audinot-Bouchez, Valérie, Boutin, Jean-Albert, Lonchampt, Michel, Dacquet, Catherine, Kto

Journal:

Year:

2012

Language:

english

File:

PDF, 926 KB

english, 2012

15

Genomic organization and characterization of splice variants of the human histamine H3 receptor

COGÉ, Francis, GUÉNIN, Sophie-Pénélope, AUDINOT, Valérie, RENOUARD-TRY, Anne, BEAUVERGER, Philippe, MACIA, Christelle, OUVRY, Christine, NAGEL, Nadine, RIQUE, Hervé, BOUTIN, Jean A., GALIZZI, Jean-Pie

Journal:

Biochemical Journal

Year:

2001

Language:

english

File:

PDF, 351 KB

english, 2001

16

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II

Sophie Durieux, Angéline Chanu, Christophe Bochu, Valérie Audinot, Sophie Coumailleau, Jean A. Boutin, Philippe Delagrange, Daniel H. Caignard, Caroline Bennejean, Pierre Renard, Daniel Lesieur, Pasca

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 380 KB

english, 2009

17

Design and Synthesis of Naphthalenic Dimers as Selective MT1 Melatoninergic Ligands

Descamps-François, Carole, Yous, Saïd, Chavatte, Philippe, Audinot, Valérie, Bonnaud, Anne, Boutin, Jean A., Delagrange, Philippe, Bennejean, Caroline, Renard, Pierre, Lesieur, Daniel

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 47 KB

english, 2003

18

Modulation of mesolimbic dopamine release by the selective dopamine D3 receptor antagonist, (+)-S 14297

Jean-Michel Rivet, Valérie Audinot, Alain Gobert, Jean-Louis Peglion, Mark J. Millan

Journal:

European Journal of Pharmacology

Year:

1994

Language:

english

File:

PDF, 264 KB

english, 1994

19

SVK14 cells express an MCH binding site different from the MCH1 or MCH2 receptor

Valérie Audinot, Chantal Lahaye, Thomas Suply, Carole Rovère-Jovène, Marianne Rodriguez, Jean-Paul Nicolas, Philippe Beauverger, Bruno Cardinaud, Jean-Pierre Galizzi, Jean-Luc Fauchère, Jean-Louis Nah

Journal:

Biochemical and Biophysical Research Communications

Year:

2002

Language:

english

File:

PDF, 155 KB

english, 2002

20

Noradrenaline and adrenaline are high affinity agonists at dopamine D4 receptors

Adrian Newman-Tancredi, Valérie Audinot-Bouchez, Alain Gobert, Mark J Millan

Journal:

European Journal of Pharmacology

Year:

1997

Language:

english

File:

PDF, 88 KB

english, 1997

21

Récepteurs couplés aux protéines G

Bril, Antoine, Combettes, Murielle, Audinot, Valérie

Journal:

médecine/sciences

Year:

2012

Language:

french

File:

PDF, 453 KB

french, 2012

22

Molecular cloning and pharmacological characterization of rat melatonin MT1 and MT2 receptors

Valérie Audinot, Anne Bonnaud, Line Grandcolas, Marianne Rodriguez, Nadine Nagel, Jean-Pierre Galizzi, Ales Balik, Sophie Messager, David G. Hazlerigg, Perry Barrett, Philippe Delagrange, Jean A. Bout

Journal:

Biochemical Pharmacology

Year:

2008

Language:

english

File:

PDF, 1.20 MB

english, 2008

23

Constitutive activity at serotonin 5-HT1D receptors: detection by homologous GTPγS versus [35S]-GTPγS binding isotherms

Valérie Audinot, Adrian Newman-Tancredi, Mark J. Millan

Journal:

Neuropharmacology

Year:

2001

Language:

english

File:

PDF, 130 KB

english, 2001

24

Agonist and antagonist actions of yohimbine as compared to fluparoxan at α2-adrenergic receptors (AR)s, serotonin (5-HT)1A, 5-HT1B, 5-HT1D and dopamine D2 and D3 receptors. Significance for the modulation of frontocortical monoaminergic transmission and depressive states

Mark J. Millan, Adrian Newman-Tancredi, Valérie Audinot, Didier Cussac, Françoise Lejeune, Jean-Paul Nicolas, Francis Cogé, Jean-Pierre Galizzi, Jean A. Boutin, Jean-Michel Rivet, Anne Dekeyne, Alain

Journal:

Year:

2000

Language:

english

File:

PDF, 340 KB

english, 2000

25

Novel benzopyrano[3,4-c]pyrrole derivatives as potent and selective dopamine D3 receptor antagonists

Thierry Dubuffet, Adrian Newman-Tancredi, Didier Cussac, Valerie Audinot, Annie Loutz, Mark J. Millan, Gilbert Lavielle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 269 KB

english, 1999

26

Alternative Etching for Improved Cu-rich CuInSe2 Solar Cells

Deprédurand, Valérie, Bertram, Tobias, Thévenin, Maxime, Valle, Nathalie, Audinot, Jean-Nicolas, Siebentritt, Susanne

Journal:

MRS Proceedings

Year:

2015

File:

PDF, 529 KB

2015

27

4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part I: Synthesis and pharmacological evaluation

Cécile Parmenon, Jérôme Guillard, Daniel-Henri Caignard, Nathalie Hennuyer, Bart Staels, Valérie Audinot-Bouchez, Jean-Albert Boutin, Catherine Dacquet, Alain Ktorza, Marie-Claude Viaud-Massuard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 182 KB

english, 2008

28

Potential Antidepressants Displayed Combined α2-Adrenoceptor Antagonist and Monoamine Uptake Inhibitor Properties

Cordi, Alex A., Berque-Bestel, Isabelle, Persigand, Thierry, Lacoste, Jean-Michel, Newman-Tancredi, Adrian, Audinot, Valerie, Millan, Mark J.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 408 KB

english, 2001

29

Preparation of 4-azaindole and 7-azaindole dimers with a bisalkoxyalkyl spacer in order to preferentially target melatonin MT1 receptors over melatonin MT2 receptors

Carlos Larraya, Jérôme Guillard, Pierre Renard, Valérie Audinot, Jean A Boutin, Philippe Delagrange, Caroline Bennejean, Marie-Claude Viaud-Massuard

Journal:

European Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 332 KB

english, 2004

30

Melanin-concentrating hormone and its receptors: state of the art

Boutin, Jean A, Suply, Thomas, Audinot, Valérie, Rodriguez, Marianne, Beauverger, Philippe, Nicolas, Jean-Paul, Galizzi, Jean-Pierre, Fauchère, Jean-Luc

Journal:

Canadian Journal of Physiology and Pharmacology

Year:

2002

File:

PDF, 1.09 MB

2002

31

Synthesis and Biological Evaluation of a New Benzofuran Analogue of 8-HETE

Renard, Pierre, Caignard, Daniel-Henri, Dacquet, Catherine, Boutin, Jean, Chomarat, Pascale, Audinot-Bouchez, Valerie, Gree, Rene, Mosset, Paul, Caijo, Frederic

Journal:

Letters in Organic Chemistry

Year:

2006

Language:

english

File:

PDF, 67 KB

english, 2006

32

New selective ligands of human cloned melatonin MT1and MT2receptors

Valérie Audinot, François Mailliet, Chantal Lahaye-Brasseur, Anne Bonnaud, Aude Le Gall, Christophe Amossé, Sandra Dromaint, Marianne Rodriguez, Nadine Nagel, Jean-Pierre Galizzi, Benoît Malpaux, Géra

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2003

Language:

english

File:

PDF, 233 KB

english, 2003

33

Genomic organization and characterization of splice variants of the human histamine H3 receptor

COGÉ, Francis, GUÉNIN, Sophie-Pénélope, AUDINOT, Valérie, RENOUARD-TRY, Anne, BEAUVERGER, Philippe, MACIA, Christelle, OUVRY, Christine, NAGEL, Nadine, RIQUE, Hervé, BOUTIN, Jean A., GALIZZI, Jean-Pie

Journal:

Biochemical Journal

Year:

2001

Language:

english

File:

PDF, 351 KB

english, 2001

34

New ligands at the melatonin binding site MT3

Marie-Françoise Boussard, Sandrine Truche, Anne Rousseau-Rojas, Sylvie Briss, Sophie Descamps, Monique Droual, Michel Wierzbicki, Gilles Ferry, Valérie Audinot, Philippe Delagrange, Jean A. Boutin

Journal:

European Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 539 KB

english, 2006

35

Synthesis of New Carbo- and Heterocyclic Analogues of 8-HETE and Evaluation of Their Activity Towards the PPARs.

Frederic Caijo, Paul Mosset, Rene Gree, Valerie Audinot-Bouchez, Jean Boutin, Pierre Renard, Daniel-Henri Caignard, Catherine Dacquet

Journal:

Year:

2006

File:

PDF, 24 KB

2006

36

Clozapine inhibits serotoninergic transmission by an action at α1-adrenoceptors not at 5-HT1A receptors

Françoise Lejeune, Valérie Audinot, Alain Gobert, Jean-Michel Rivet, Michael Spedding, Mark J. Millan

Journal:

European Journal of Pharmacology

Year:

1994

Language:

english

File:

PDF, 398 KB

english, 1994

37

S38151 [p-guanidinobenzoyl-[Des-Gly10]-MCH(7-17)] is a potent and selective antagonist at the MCH1 receptor and has anti-feeding properties in vivo

Valérie Audinot, Odile Della Zuana, Nelly Fabry, Christine Ouvry, Olivier Nosjean, Jean-Michel Henlin, Jean-Luc Fauchère, Jean A. Boutin

Journal:

Year:

2009

Language:

english

File:

PDF, 862 KB

english, 2009

38

Molecular identification of the long isoform of the human neuropeptide Y Y5 receptor and pharmacological comparison with the short Y5 receptor isoform

RODRIGUEZ, Marianne, AUDINOT, Valérie, DROMAINT, Sandra, MACIA, Christelle, LAMAMY, Véronique, BEAUVERGER, Philippe, RIQUE, Hervé, IMBERT, Jérôme, NICOLAS, Jean Paul, BOUTIN, Jean A., GALIZZI, Jean Pi

Journal:

Biochemical Journal

Year:

2003

Language:

english

File:

PDF, 206 KB

english, 2003

39

Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARγ agonists

Elodie Blanc-Delmas, Nicolas Lebegue, Valérie Wallez, Véronique Leclerc, Saïd Yous, Pascal Carato, Amaury Farce, Caroline Bennejean, Pierre Renard, Daniel-Henri Caignard, Valérie Audinot-Bouchez, Pasc

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 421 KB

english, 2006

40

Tetracyclic analogues of [+]-S 14297: Synthesis and determination of affinity and selectivity at cloned human dopamine D3 vs D2 receptors

Jean-Louis Peglion, Joël Vian, Bertrand Goument, Nicole Despaux, Valérie Audinot, Mark J. Millan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 330 KB

english, 1997

41

Design and synthesis of 3-phenyl tetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands

Saı̈d Yous, Sophie Durieux-Poissonnier, Emmanuelle Lipka-Belloli, Halim Guelzim, Christophe Bochu, Valérie Audinot, Jean A Boutin, Philippe Delagrange, Caroline Bennejean, Pierre Renard, Daniel Lesieu

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 177 KB

english, 2003

42

Molecular tools to study melatonin pathways and actions

Jean A. Boutin, Valérie Audinot, Gilles Ferry, Philippe Delagrange

Journal:

Trends in Pharmacological Sciences

Year:

2005

Language:

english

File:

PDF, 312 KB

english, 2005

43

Characterization of Potent and Selective Antagonists at Postsynaptic 5-HT1A Receptors in a Series of N4-Substituted Arylpiperazines

Peglion, Jean-Louis, Canton, Herve, Bervoets, Karin, Audinot, Valerie, Brocco, Mauricette, Gobert, Alain, Le Marouille-Girardon, Sylvie, Millan, Mark J.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 1.37 MB

english, 1995

44

Peripheral injections of melanin-concentrating hormone receptor 1 antagonist S38151 decrease food intake and body weight in rodent obesity models

Della-Zuana, Odile, Audinot, Valérie, Levenez, Viviane, Ktorza, Alain, Presse, Françoise, Nahon, Jean-Louis, Boutin, Jean A.

Journal:

Frontiers in Endocrinology

Year:

2012

Language:

english

File:

PDF, 3.68 MB

english, 2012

45

Functional characterization of human neuropeptide Y receptor subtype five specific antagonists using a luciferase reporter gene assay

Philippe Beauverger, Marianne Rodriguez, Jean-Paul Nicolas, Valérie Audinot, Véronique Lamamy, Sandra Dromaint, Nadine Nagel, Christelle Macia, Odile Léopold, Jean-Pierre Galizzi, Daniel-Henri Caignar

Journal:

Cellular Signalling

Year:

2005

Language:

english

File:

PDF, 488 KB

english, 2005

46

Benzamides derived from 1,2-diaminocyclopropane as novel ligands for human D2 and D3 dopamine receptors

Donglai Yang, Slaheddine Kefi, Valérie Audinot, Mark-J. Millan, Michel Langlois

Journal:

Bioorganic & Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 201 KB

english, 2000

47

Mechanistic characterization of S 38093, a novel inverse agonist at histamine H3 receptors

Sors, Aurore, Panayi, Fany, Bert, Lionel, Favale, Dominique, Nosjean, Olivier, Audinot, Valérie, Arrang, Jean-Michel, Buisson, Bruno, Steidl, Esther, Delbos, Jean-Marie, Huhtala, Tuulia, Kontkanen, Ou

Journal:

European Journal of Pharmacology

Year:

2017

Language:

english

File:

PDF, 1.20 MB

english, 2017

48

Synthesis of Aromatic Analogs of 8(S)-HETE and Their Biological Evaluation as Activators of the PPAR Nuclear Receptors

Frédéric Caijo, Paul Mosset, René Grée, Valérie Audinot-Bouchez, Jean Boutin, Pierre Renard, Daniel-Henri Caignard, Catherine Dacquet

Journal:

European Journal of Organic Chemistry

Year:

2006

Language:

english

File:

PDF, 293 KB

english, 2006

49

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT1 melatoninergic ligands

Christophe Mésangeau, Basile Pérès, Carole Descamps-François, Philippe Chavatte, Valérie Audinot, Sophie Coumailleau, Jean A. Boutin, Philippe Delagrange, Caroline Bennejean, Pierre Renard, Daniel H.

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 719 KB

english, 2010

50

Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPγS binding study

Adrian Newman-Tancredi, Samantha Gavaudan, Caroline Conte, Christine Chaput, Manuelle Touzard, Laurence Verrièle, Valerie Audinot, Mark J Millan

Journal:

European Journal of Pharmacology

Year:

1998

Language:

english

File:

PDF, 254 KB

english, 1998

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